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02690 CONTEMPORAY MATERIAL CONCEPTS FOR THE NEXT GENERATION MICROBICIDE VEHICLES Kiser, Patrick In the last 20 years there has been a revolution in understanding the underlying principles of bioresponsive materials for drug delivery and formulation science. These principles, developed by material scientists and pharmaceutics researchers, are now being applied to first generation microbicides, e.g. in the pegylated active ingredients such as PEG-cyanovirin and in thermo-gelling systems. We are developing a number of approaches to create novel bioresponsive materials and formulations for drug delivery in the vagina that are potential prototypes for 2nd and 3rd generation microbicidal formulations. Our approach is to engineer new materials that are designed to undergo changes in their properties in response to interactions with biological triggers that exist in the vagina, including pH, temperature and shear fields. By utilizing contemporary materials we are able to affect significant changes in rheological and other salient physico-chemical properties in response to these triggers. We hypothesize that these changes will enhance the bioactivity of the active ingredient and the carrier, as well as the biodistribution in the vagina. We are currently designing and testing several polymer systems which leverage these bioresponsive signals to create carriers that in themselves are active, and/or modify the properties of the active pharmaceutical in the vagina. Assistant Professor, Patrick, Kiser |
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