![]() |
![]() |
||||||||||||
|
02664 DEVELOPMENT OF MICROBICIDE VEHICLES: SELECTION LINKED TO PROPERTIES GOVERNING VAGINAL DEPLOYMENT Owen*, Derek A set of 12 prototype gels was created for potential use as vehicles for new microbicides under development. These gels were of four types: cellulose/polymer-cationic (A), cellulose-nonionic (B), block copolymer-nonionic (C), and poly acrylic acid/cellulose-anionic (D). The different combinations of molecular composition were intended to produce gels with different biophysical properties that govern vaginal distribution and retention (deployment). Variation of these properties was intended to enable testing of hypotheses regarding how different combinations of gel characteristics lead to better or worse deployment. The rheological properties of these gels were studied for whole gels and after dissolution with vaginal fluid and semen simulants. The gels exhibited a wide range of rheological properties. For example, the gels of type C and D exhibited yield stresses while gels of type A and B did not. The four types of gels also exhibited different viscosities and shear thinning behavior. Dissolution studies indicated substantial differences in the propensity of the gel layer to be washed off by the simulants. Some gels swelled while the gel layer remained intact while others rapidly dissolved with loss of the gel layer. The results suggest significant differences in the vaginal deployment of the test gels. (Sponsored by NIH Grant # U19AI051650-02 to Biosyn Inc and, NIH Grant # AI48103 to Duke University). Assistant Research Professor Derek Owen |
|||||||||||||