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02387 EUROPEAN MICROBICIDES PROJECT Kelly, Charles* The European Microbicides Project (EMPRO) is a consortium of 35 principal investigators from 29 institutions or SMEs that has been funded by the European Union as part of the Sixth Framework Programme in the area Confronting the major communicable diseases linked to poverty. The programme aims to develop new topical microbicides, with defined molecular targets, that block entry of HIV at mucosal sites with the aim of establishing a pipeline of candidate microbicides while taking selected microbicides through Phase I clinical trials. Members of the consortium have expertise in analyses and design of molecular structure, investigation of mechanisms of HIV infection at mucosal sites, testing efficacy in animal models, methods for large-scale production of microbicides and the conduct of clinical trials. Novel molecules and combinatorial peptide, polypeptide and oligosaccharide libraries will be screened for inhibitors that are specifically targeted to viral envelope proteins or host receptors. Microbicidal efficacy and effect on normal microbial flora of inhibitors will be tested in vitro. The most promising candidate microbicides will be formulated and tested in animal models. The developmental process for candidate agents will be target-driven according to a preclinical selection algorithm designed to fast track the most promising candidates and/or combination. Emphasis will be placed on development of compounds demonstrating synergistic activity either with others from this programme or with first generation compounds developed by other groups that are further ahead in the developmental process. As well as identifying novel candidate microbicides, the programme should provide a rational basis for the design of 2nd or 3rd generation microbicides. Professor Charles Kelly |
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