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02230 IN VITRO SAFETY EVALUATION OF A COMBINATIONAL MICROBICIDE CANDIDATE, PL40, Ben, Kunlong1 In order to evaluate the safety of a combinational microbicide candidate, PL40, which is composed of PS 20 and LN 43, their cytotoxicities to human cervical cancer cell lines ME-180 and HeLa, and to primary foreskin keratinocytes (PFK) were detected by MTT assay. The activity of anti-Lactobacillus debrueckii, a member of normal vaginal flora, was measured by microdilution method. Inhibition concentrations (IC50s) of PS20 were 3.2 mg/ml for ME-180, 2 mg/ml for HeLa, 1.5mg/ml for PFK cells, and IC50s of LN43 were 4.6 mM, 4.3 mM and 1.2 mM, respectively. All IC50s are several hundreds times of effective concentrations (EC50s) of both compounds for inhibiting HIV-1 infection. The minimal inhibition concentrations (MICs) of both PS20 and LN43 for Lactobacillus debrueckii were more than 20 mg/ml, and are almost 1000 times of EC50s of the compounds for their anti-HIV-1 activities. These results suggest that the components of PL40 have very low toxicity to cells of human genital tracts as well as to normal bacteria in the above in vitro tests. Professor, General manager, Kunlong Ben |
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