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02655 VAGINAL TENOFOVIR GEL TOLERABILITY IN HIV-UNINFECTED WOMEN AND ABSTINENT HIV-INFECTED WOMEN:HPTN 050 Maslankowski, Lisa1 Objective: To establish the highest tolerated dose and frequency of once daily or twice daily 0.3% and 1% Tenofovir (PMPA) vaginal gel in abstinent HIV-uninfected (HIV-) women and to evaluate this dose in sexually active HIV- women and abstinent HIV-infected (HIV+) women. To describe systemic pharmacokinetics (PK) of Tenofovir vaginal gel in a subset of participants. Methods: Safety labs and pelvic exams were completed at screening, enrollment, Day 2-3, Day 7 and Day 14 visits with colposcopy at enrollment and the Day 14 visit. Women used study product for 14 consecutive days. PK samples were collected after a single application and on Day 13. Results: Seventy-two women were enrolled. Since 1% BID was as well tolerated as lower doses/frequencies, it was evaluated in the sexually active HIV- and abstinent HIV+ cohorts. Adverse events (AEs) were reported in 66 women. Most were mild genital AEs such as erythema(n=15), ecchymosis/petechiae(n=13), or pruritis (n=12). One severe adverse event (abdominal pain) possibly related to product was reported. Ten of 19 women in the PK subset had low but detectable tenofovir serum concentrations (lower level of quantification=2.99 ng/ml, Cmax ranged from 3.01 25.83). Conclusion: Tenofovir (PMPA) vaginal gel 1% BID is well tolerated in HIV- women and abstinent HIV+ women with minimal systemic absorption. Evaluation of sexually active HIV+ women is underway. Phase II extended safety and effectiveness testing is planned. Dr. Lisa Maslankowski |
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